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- Total synthesis of mannopeptimycin β via βhydroxyenduracididine ligation. Wang, J.; Lin, D.; Liu, M.; Liu, H.; Li, X.* J. Am. Chem. Soc. 2021, 143, 12784.
- Chemical Synthesis and Biological Evaluation of Adiponectin Collagenous Domain Glycoforms. Wu, H.; Zhang, Y.; Li, Y.; Xu, J.; Wang, Y.*; Li, X.* J. Am. Chem. Soc. 2021, 143, 7808-7818.
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- Total Synthesis of Malacidin A by β-Hydroxyaspartic Acid Ligation Mediated Cyclization and Absolute Structure Establishment. Sun, Z.; Shang, Z.; Forelli, N.; Po, K. H. Y.; Chen, S.; Brady, S. F.*; Li X.* Angew. Chem. Int. Ed. 2020, 15, 19868- 19872.
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